SCHEMBL7364226

SCHEMBL7364226

CCOc1ccc(NC(=O)c2c[nH]c3c2C(=O)CCCC3)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.42
DHODH Q02127 3/20 0.39
NR4A2 P43354 2/20 0.39
MRGPRX1 Q96LB2 1/20 0.39
POLB P06746 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
MCOLN3 Q8TDD5 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPY2R P49146 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7363435 0.98 DHODH (0.41) TP53DHODHNR4A2MRGPRX1POLB
SCHEMBL6095595 0.89 DHODH (0.40) TP53DHODHNR4A2HTTSCN8A
SCHEMBL7359461 0.89 DHODH (0.44) DHODHNR4A2MAPTMEN1LMNA
SCHEMBL6092670 0.87 DHODH (0.42) DHODHNR4A2LMNAHTTSCN8A
SCHEMBL7400116 0.87 DHODH (0.47) DHODHNR4A2POLBMAPTNPC1
SCHEMBL6094311 0.86 DHODH (0.43) TP53DHODHNR4A2MAPTHTT
SCHEMBL7397673 0.85 POLB (0.40) TP53DHODHNR4A2MRGPRX1POLB
SCHEMBL6773568 0.85 L3MBTL1 (0.41) TP53MRGPRX1POLBL3MBTL1ATM
SCHEMBL7363099 0.85 DHODH (0.46) DHODHNR4A2POLBMAPTLMNA
SCHEMBL6776660 0.85 MAPT (0.40) TP53MRGPRX1POLBL3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO claimed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO claimed
WO-1998002420-A9 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS 1998-04-23 WO disclosed
WO-1998002420-A1 CERTAIN FUSED PYRROLECARBOXANILIDES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1998-01-22 WO disclosed