SCHEMBL7364696

SCHEMBL7364696

CCOC(=O)[C@@H](CCc1ccccc1)[C@@]1(C(=O)O)CCCN1C(=O)[C@H](C)N

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 12/20 0.44
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
ABCB11 O95342 1/20 0.40
POLB P06746 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL7318816 0.95 SMN1; SMN2 (0.47) ACELMNASMN1; SMN2ABCB11POLB
SCHEMBL9394613 0.89 ACE (0.40) ACEALDH1A1
SCHEMBL7266941 0.87 ACE (0.42) ACELMNAPOLBALDH1A1
SCHEMBL8715043 0.78 ACE (0.49) ACELMNASMN1; SMN2ABCB11MEN1
SCHEMBL5551908 0.76 DPP8 (0.40) ACE
SCHEMBL10883512 0.75 DPP7 (0.39) ACE
SCHEMBL8568423 0.75 ACE (0.45) ACELMNASMN1; SMN2POLBALDH1A1
SCHEMBL10696084 0.75 ACE (0.45) ACELMNASMN1; SMN2POLBALDH1A1
SCHEMBL649164 0.74 DPP8 (0.43) ACE
SCHEMBL5552493 0.74 DPP8 (0.43) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523449-B1 Reductive amination of an aminoacid or an aminoacid derivative with an alpha-keto acid or an alpha-keto acid derivative DEGUSSA (DE) 1996-05-15 EP disclosed
EP-0523449-A2 Reductive amination of an aminoacid or an aminoacid derivative with an alpha-keto acid or an alpha-keto acid derivative DEGUSSA AG (DE) 1993-01-20 EP disclosed
EP-0012401-A1 Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them MERCK & CO. INC. (US) 1980-06-25 EP disclosed