SCHEMBL7364823

SCHEMBL7364823

COc1cc(NCc2ccccc2OCCCCN2CCN(C(C)=O)CC2)ccc1C(=O)N1CCCCc2cc(Cl)ccc21

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 12/20 0.48
TP53 P04637 2/20 0.40
TSHR P16473 1/20 0.40
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4683205 0.89 AVPR2 (0.52) AVPR2TP53
SCHEMBL7348955 0.83 AVPR2 (0.55) AVPR2TP53
SCHEMBL4687327 0.79 AVPR2 (0.55) AVPR2TP53
SCHEMBL8632240 0.70 AVPR2 (0.44) AVPR2
SCHEMBL8630825 0.70 AVPR2 (0.40) AVPR2
Hydrochloric Acid SCHEMBL8628767 0.69 AVPR2 (0.47) AVPR2TP53TSHR
SCHEMBL7017339 0.69 AVPR2 (0.46) AVPR2
SCHEMBL4685041 0.68 CHRM5 (0.44) AVPR2TP53
SCHEMBL4687283 0.68 AVPR2 (0.51) AVPR2
Hydrochloric Acid SCHEMBL7338452 0.68 AVPR2 (0.57) AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514667-A1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-25 EP disclosed