SCHEMBL7364910

SCHEMBL7364910

CCOC(=O)c1ccc(C)nc1C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA7 P43166 2/20 0.45
CA9 Q16790 2/20 0.45
CA14 Q9ULX7 2/20 0.45
CYP1A2 P05177 1/20 0.45
ALDH1A1 P00352 7/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4E B2RXH2 4/20 0.42
ALOX15 P16050 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CDC25B P30305 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5078941 0.86 CA12 (0.47) TSHRCA12CA1CA2CA7
SCHEMBL5079690 0.84 TSHR (0.46) TSHRMEN1KMT2ACA12CA1
SCHEMBL30040951 0.81 KDM4E (0.51) TSHRMEN1KMT2ACA12CA1
SCHEMBL9355979 0.80 TSHR (0.55) TSHRMEN1KMT2ACA12CA1
SCHEMBL5664007 0.80 KDM4E (0.57) TSHRMEN1KMT2ACA12CA1
SCHEMBL16828808 0.78 MEN1 (0.55) TSHRMEN1KMT2ACA12CA1
SCHEMBL9308330 0.78 TSHR (0.53) TSHRMEN1KMT2ACA12CA1
SCHEMBL7354531 0.78 TSHR (0.53) TSHRMEN1KMT2ACA12CA1
SCHEMBL18882780 0.78 SORT1 (0.43) MEN1KMT2ACYP1A2ALDH1A1SMN1; SMN2
SCHEMBL26713458 0.78 SMN1; SMN2 (0.41) ALDH1A1HSD17B10KDM4ESMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0805681-A4 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-05-06 EP disclosed
EP-0805681-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1997-11-12 EP disclosed
WO-1996022775-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-08-01 WO disclosed