SCHEMBL7365042

SCHEMBL7365042

CC(C)Cc1nc(C2CCCN(C)C2)oc1C(=O)CNC(=O)CC(C)(C)CC(N)=O

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
ASAH1 Q13510 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359424 0.86 ERCC1 (0.35) ERCC1ERCC4ASAH1
SCHEMBL6803756 0.82 ERCC1 (0.35) ERCC1ERCC4ASAH1
SCHEMBL6803750 0.82 ERCC1 (0.33) ERCC1ERCC4ASAH1
SCHEMBL6800978 0.81 ASAH1 (0.36) ERCC1ERCC4ASAH1
SCHEMBL6800971 0.80 ERCC1 (0.34) ERCC1ERCC4ASAH1
SCHEMBL6807167 0.66 ERCC1 (0.34) ERCC1ERCC4ASAH1
SCHEMBL7366743 0.64 LMNA (0.41)
SCHEMBL6802745 0.64 AXL (0.32)
Oxalic Acid SCHEMBL10418863 0.54 HSD11B1 (0.42)
SCHEMBL13722060 0.53 EPHA2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed