SCHEMBL7365503

SCHEMBL7365503

COC(=O)C[C@H]1C(=O)N(CC(=O)O)CCN1C(=O)C(CC(=O)N1CCN(c2ccncc2)CC1)Cc1ccc(OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.44
ITGA2B P08514 7/20 0.44
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
GFER P55789 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.36
P2RX7 Q99572 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933354 1.00 ITGB3 (0.44) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7367151 0.93 GFER (0.38) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7367152 0.93 GFER (0.38) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7365965 0.89 ITGB3 (0.43) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7365953 0.89 ITGB3 (0.43) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7365958 0.89 ITGB3 (0.43) ITGB3ITGA2BALDH1A1GAAHSD17B10
Trifluoroacetic Acid SCHEMBL7924758 0.86 ITGB3 (0.40) ITGB3ITGA2BALDH1A1GAAHSD17B10
Trifluoroacetic Acid SCHEMBL7369430 0.86 ITGB3 (0.40) ITGB3ITGA2BALDH1A1GAAHSD17B10
SCHEMBL7370702 0.85 ITGB3 (0.46) ITGB3ITGA2BTSHR
SCHEMBL7935145 0.85 ITGB3 (0.46) ITGB3ITGA2BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242600-B1 ANTIISCHEMIC AGENTS, ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-05 US disclosed
EP-0970071-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-12 EP disclosed
WO-1998039324-A1 2-PEPERAZINONE-1-ACETIC ACID DERIVATIVES AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-11 WO disclosed