SCHEMBL7365926

SCHEMBL7365926

O=C/C=C(/Cl)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 4/20 0.44
MAPK1 P28482 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CES1 P23141 5/20 0.40
CES2 O00748 4/20 0.40
TSHR P16473 2/20 0.40
DAO P14920 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
TRPA1 O75762 1/20 0.38
GSK3B P49841 1/20 0.38
HIF1A Q16665 1/20 0.38
AKT1 P31749 1/20 0.38
CA2 P00918 3/20 0.37
CYP3A4 P08684 2/20 0.37
MAPT P10636 2/20 0.37
CA4 P22748 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL560304 1.00 MEN1 (0.46) MEN1KMT2AALDH1A1MAPK1TDP1
SCHEMBL2098803 1.00 MEN1 (0.46) MEN1KMT2AALDH1A1MAPK1TDP1
SCHEMBL18690045 0.88 MEN1 (0.39) MEN1KMT2AALDH1A1MAPK1TDP1
SCHEMBL26490231 0.81 PARP10 (0.57) MEN1KMT2AALDH1A1TDP1SMN1; SMN2
SCHEMBL23275547 0.81 PARP10 (0.57) MEN1KMT2AALDH1A1TDP1SMN1; SMN2
SCHEMBL2559260 0.79 CES2 (0.46) ALDH1A1MAPK1CES1CES2TSHR
SCHEMBL2559262 0.79 CES2 (0.46) ALDH1A1MAPK1CES1CES2TSHR
SCHEMBL8338715 0.79 CES2 (0.46) ALDH1A1MAPK1CES1CES2TSHR
SCHEMBL11172576 0.78 AKR1C3 (0.57) ALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL11172580 0.78 AKR1C3 (0.57) ALDH1A1SMN1; SMN2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992577-A Preparation of 3-vinyl-substituted 2,2-dimethylcyclopropane-1-carboxylic acids and esters and intermediates therefor BAYER AKTIENGESELLSCHAFT (DE) 1991-02-12 US disclosed
US-4755599-A 3-phenyl-2-propeneamine derivatives, their preparation and composition containing them RHONE-POULENC SANTE (FR) 1988-07-05 US disclosed
US-4686309-A ANTIDEPRESSANTS RHONE-POULENC SANTE (FR) 1987-08-11 US disclosed
EP-0095047-B1 PROCESS FOR THE PREPARATION OF 3-VINYL-SUBSTITUTED 2,2-DIMETHYL-CYCLOPROPANE-1-CARBOXYLIC ACIDS OR THEIR ESTERS, AND INTERMEDIATE PRODUCTS THEREFOR BAYER AG (DE) 1985-11-27 EP disclosed
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed
US-4221895-A POLYESTER, POLYSULFONATE, OR POLYSULFINATE THE DOW CHEMICAL COMPANY (US) 1980-09-09 US disclosed