SCHEMBL7366426

SCHEMBL7366426

COc1ccc(C#N)c(CO)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.50
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
MAOB P27338 1/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 1/20 0.45
KDM4E B2RXH2 4/20 0.43
AR P10275 3/20 0.43
ALDH1A1 P00352 3/20 0.43
MAOA P21397 1/20 0.43
PGR P06401 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GLA P06280 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CLK1 P49759 1/20 0.41
CASP7 P55210 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672598 0.87 NPC1 (0.47) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL7320659 0.87 PGR (0.56) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL13652097 0.84 NOS2 (0.51) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL16958190 0.83 GLA (0.47) NPC1RAB9AMAOBHSD17B10TP53
SCHEMBL3045111 0.82 NOS2 (0.50) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL8176765 0.82 NOS2 (0.50) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL7663985 0.82 NOS2 (0.50) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL3054041 0.82 NOS2 (0.50) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL7366242 0.82 NOS2 (0.53) NOS2NPC1RAB9AMAOBHSD17B10
SCHEMBL16313416 0.81 NOS2 (0.49) NOS2NPC1RAB9AMAOBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
EP-1259506-A1 PYRAZINONE THROMBIN INHIBITORS Merck & Co., Inc. (US) 2002-11-27 EP disclosed
US-6476021-B1 Compounds having cGMP-PDE inhibitory effect MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-11-05 US disclosed
US-6387911-B1 Pyrazinone thrombin inhibitors MERCK & CO., INC. 2002-05-14 US disclosed
WO-2001038323-A1 PYRAZINONE THROMBIN INHIBITORS MERCK & CO., INC. (US) 2001-05-31 WO disclosed
EP-1048666-A1 NOVEL COMPOUNDS HAVING cGMP-PDE INHIBITORY EFFECT MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2000-11-02 EP disclosed