SCHEMBL7366432

SCHEMBL7366432

CC(C)(C)OC(=O)Nc1ccc2cn[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.57
CYP1A2 P05177 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2D6 P10635 2/20 0.57
CYP2C9 P11712 2/20 0.57
HIF1A Q16665 2/20 0.57
HSD17B10 Q99714 2/20 0.57
CYP2C19 P33261 1/20 0.57
PHLPP2 Q6ZVD8 1/20 0.57
KDM4E B2RXH2 10/20 0.55
MAPT P10636 9/20 0.55
MAP4K4 O95819 1/20 0.54
CLK2 P49760 1/20 0.54
DYRK1A Q13627 1/20 0.54
SRPK1 Q96SB4 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
HPGD P15428 3/20 0.53
F2 P00734 2/20 0.53
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31467439 1.00 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL625972 0.89 ROCK2 (0.66) MAP4K4CLK2DYRK1ACLK4RAB9A
SCHEMBL15764690 0.82 NPC1 (0.68) MAP4K4CLK2DYRK1ACLK4RAB9A
SCHEMBL22590423 0.82 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3720338 0.81 GSK3B (0.56)
SCHEMBL3720334 0.81 GSK3B (0.56)
SCHEMBL3720332 0.81 GSK3B (0.56)
SCHEMBL3716869 0.80 GSK3B (0.48)
SCHEMBL3716865 0.80 GSK3B (0.48)
SCHEMBL3716868 0.80 GSK3B (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023122756-A2 ULK1 AND ULK2 INHIBITORS BOARD OF TRUSTEES OF MICHIGAN STATE UNIVERSITY (US) 2023-06-29 WO disclosed
EP-1019045-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2002-07-03 EP disclosed
EP-1019045-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-19 EP disclosed
WO-1999000128-A9 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 1999-08-05 WO disclosed
WO-1999000128-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed