SCHEMBL7366465

SCHEMBL7366465

CCCCN(C=CC(=O)c1cccnc1)CCCC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.50
MAPT P10636 4/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 5/20 0.49
CYP1A1 P04798 4/20 0.49
CYP1B1 Q16678 4/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2D6 P10635 3/20 0.49
LMNA P02545 3/20 0.48
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
GPR52 Q9Y2T5 1/20 0.47
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10938347 1.00 MAPK1 (0.52) MAPK1NPSR1L3MBTL1MAPTKMT2A
SCHEMBL7368742 0.86 MAPK1 (0.60) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL7368740 0.86 MAPK1 (0.60) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL30269691 0.78 HTT (0.65) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL1643 0.78 HTT (0.65) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL29364482 0.78 HTT (0.65) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL1218 0.78 HTT (0.65) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL9486033 0.78 HTT (0.65) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL3262039 0.78 CYP1A1 (0.51) MAPK1NPSR1MAPTKMT2AMEN1
SCHEMBL3262042 0.78 CYP1A1 (0.51) MAPK1NPSR1MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed