SCHEMBL7368740

SCHEMBL7368740

CCN(/C=C/C(=O)c1cccnc1)CC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
CYP1A1 P04798 6/20 0.54
CYP1A2 P05177 6/20 0.54
CYP1B1 Q16678 6/20 0.54
CYP3A4 P08684 4/20 0.54
CYP2D6 P10635 4/20 0.54
MAPT P10636 3/20 0.53
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.53
GPR52 Q9Y2T5 1/20 0.51
HTT P42858 1/20 0.50
ALDH1A1 P00352 2/20 0.49
LMNA P02545 2/20 0.49
HPGD P15428 1/20 0.49
APP P05067 1/20 0.48
GSK3B P49841 1/20 0.48
KDM4E B2RXH2 1/20 0.48
CAPN1 P07384 1/20 0.47
CTSL P07711 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368742 1.00 MAPK1 (0.60) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL7366465 0.86 MAPK1 (0.52) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL10938347 0.86 MAPK1 (0.52) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL29364482 0.83 HTT (0.65) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL1643 0.83 HTT (0.65) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL30269691 0.83 HTT (0.65) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL9486033 0.83 HTT (0.65) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL1218 0.83 HTT (0.65) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL3262042 0.82 CYP1A1 (0.51) MAPK1NPSR1CYP1A1CYP1A2CYP1B1
SCHEMBL3262039 0.82 CYP1A1 (0.51) MAPK1NPSR1CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521422-A ANTICONVULSANT, ANTIEPILEPTIC AGENTS, SEDATIVES, MUSCLE RELAXANTS AMERICAN CYANAMID COMPANY (US) 1985-06-04 US disclosed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed