SCHEMBL7366718

SCHEMBL7366718

COC(=O)c1cccnc1Oc1ccc(C#N)cc1

nearest known ligand 0.71

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.71
ALDH1A1 P00352 1/20 0.48
RAB9A P51151 1/20 0.48
DRD1 P21728 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
GAA P10253 1/20 0.47
ROCK2 O75116 1/20 0.46
HPGD P15428 1/20 0.46
MAPK8 P45983 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL850967 0.86 ELANE (0.53) TDP1ALDH1A1GAA
SCHEMBL851191 0.85 TDP1 (0.52) TDP1ALDH1A1RAB9AGAAROCK2
SCHEMBL20818012 0.83 TDP1 (1.00) TDP1ALDH1A1RAB9AGAAMAPK8
SCHEMBL7373227 0.82 TDP1 (0.76) TDP1ALDH1A1RAB9AGAAHPGD
SCHEMBL620646 0.82 TDP1 (0.76) TDP1ALDH1A1RAB9ADRD1GAA
SCHEMBL28069342 0.82 TDP1 (0.76) TDP1ALDH1A1RAB9ADRD1GAA
SCHEMBL28734386 0.80 TDP1 (0.72) TDP1ALDH1A1RAB9ADRD1CYP1A2
SCHEMBL5749934 0.80 TDP1 (0.72) TDP1ALDH1A1RAB9ADRD1GAA
SCHEMBL620688 0.78 TDP1 (0.69) TDP1ALDH1A1RAB9ADRD1GAA
SCHEMBL10976046 0.76 TDP1 (0.67) TDP1ALDH1A1RAB9ADRD1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380218-B1 FOR THERAPY OF RESPIRATORY, ALLERGIC, AND INFLAMMATORY DISORDERS COMPRISING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ACUTE RESPIRATORY DISEASE SYNDROME, PULMONARY HYPERSENSITIVITY, AND ALLERGIC RHINITIS IN A MAMMAL PFIZER INC 2002-04-30 US disclosed
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed