SCHEMBL7366847

SCHEMBL7366847

O=C(O)COc1noc(-c2cccs2)c1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
NR1H4 Q96RI1 2/20 0.40
MAPT P10636 2/20 0.38
ALDH1A1 P00352 3/20 0.38
GLA P06280 1/20 0.38
BRCA1 P38398 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
MCL1 Q07820 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CA12 O43570 2/20 0.36
CA9 Q16790 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370266 0.80 SMN1; SMN2 (0.44) TSHRMAPTALDH1A1CYP1A2CYP2C19
SCHEMBL7374874 0.80 SMN1; SMN2 (0.41) NR1H4MAPTALDH1A1FABP3FABP4
SCHEMBL7406142 0.76 GRIA1 (0.58) CYP1A2CYP2C19SMN1; SMN2KDM4EHPGD
SCHEMBL7406133 0.76 GRIA1 (0.58) CYP1A2CYP2C19SMN1; SMN2KDM4EHPGD
SCHEMBL7367693 0.76 KDM4E (0.43) TSHRMAPTALDH1A1CYP1A2CYP2C19
SCHEMBL7373678 0.74 NPC1 (0.43) NR1H4ALDH1A1GLASMN1; SMN2KDM4E
SCHEMBL8120933 0.73 GRIN2D (0.39) MAPTALDH1A1CYP1A2CYP2C19MCL1
SCHEMBL7374568 0.71 MAPT (0.50) TSHRMAPK1MAPTALDH1A1BRCA1
SCHEMBL8120929 0.69 MCL1 (0.36) TSHRMAPTALDH1A1FABP3FABP4
SCHEMBL7406301 0.65 GRIA1 (0.44) MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994107-A1 5-Arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds H. LUNDBECK A/S (DK) 2000-04-19 EP disclosed
EP-0726896-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1996-08-21 EP disclosed
WO-1995012587-A1 5-ARYLISOXAZOL-4-YL-SUBSTITUTED 2-AMINO CARBOXYLIC ACID COMPOUNDS H. LUNDBECK A/S (DK) 1995-05-11 WO disclosed