SCHEMBL7366867

SCHEMBL7366867

Cc1cc(C)c(S(=O)(=O)[C@H](C(=O)c2nnc(CCCCNC3=NCCN3)s2)C(N)(N)C(=O)O)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.42
ITGAV P06756 7/20 0.42
ITGA2B P08514 6/20 0.42
ITGB1 P05556 1/20 0.35
CXCR4 P61073 3/20 0.34
F2 P00734 2/20 0.32
WDR5 P61964 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366861 1.00 ITGB3 (0.42) ITGB3ITGAVITGA2BITGB1CXCR4
SCHEMBL7369530 0.82 ITGB3 (0.41) ITGB3ITGAVITGA2BITGB1
SCHEMBL7369525 0.82 ITGB3 (0.41) ITGB3ITGAVITGA2BITGB1
SCHEMBL7373174 0.81 ITGB3 (0.43) ITGB3ITGAVITGA2BITGB1CXCR4
SCHEMBL7367256 0.81 F2 (0.40) ITGB3ITGAVITGA2BCXCR4F2
SCHEMBL7367251 0.81 F2 (0.40) ITGB3ITGAVITGA2BCXCR4F2
SCHEMBL7373177 0.81 ITGB3 (0.43) ITGB3ITGAVITGA2BITGB1CXCR4
SCHEMBL8176082 0.78 ITGAV (0.65) ITGB3ITGAVITGA2BITGB1
SCHEMBL7377522 0.75 ITGB3 (0.36) ITGB3ITGAVITGA2BCXCR4F2
SCHEMBL7377515 0.75 ITGB3 (0.36) ITGB3ITGAVITGA2BCXCR4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP claimed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO claimed
EP-1049693-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS $g(a) v?$g(b) 3? ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-08 EP disclosed
WO-1999026945-A1 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES AS αvβ3 ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-06-03 WO disclosed