SCHEMBL7367610

SCHEMBL7367610

CC(C(=O)O)n1ccc2cc(C#N)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.41
NPY5R Q15761 1/20 0.39
CDC7 O00311 1/20 0.39
PTGER4 P35408 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
P2RX7 Q99572 1/20 0.37
PRMT5 O14744 1/20 0.37
ENPP3 O14638 1/20 0.36
CCR9 P51686 1/20 0.36
ALB P02768 1/20 0.36
IRAK4 Q9NWZ3 3/20 0.36
ABCB1 P08183 2/20 0.36
F2 P00734 1/20 0.35
PLG P00747 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2414232 0.82 CCR9 (0.39) FFAR4NPY5RCDC7KDM4EALDH1A1
SCHEMBL3709688 0.82 CDC7 (0.43) FFAR4NPY5RCDC7KDM4EALDH1A1
SCHEMBL6258605 0.79 HTR2A (0.45) ALDH1A1PTGS2
SCHEMBL22798768 0.78 SLC6A2 (0.48) TSHRPTGS2
SCHEMBL22798937 0.78 SLC6A2 (0.48) TSHRPTGS2
SCHEMBL22798770 0.78 SLC6A2 (0.48) TSHRPTGS2
SCHEMBL16627458 0.78 NTSR1 (0.50) HTTPTGS2
SCHEMBL22798848 0.78 NTSR1 (0.50) HTTPTGS2
SCHEMBL16619844 0.78 NTSR1 (0.50) HTTPTGS2
SCHEMBL22320205 0.77 CDC7 (0.40) FFAR4NPY5RCDC7KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043257-A ANTICOAGULANT; PYRIDINE SUBSTITUTED INDAZOLE COMPOUND E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-03-28 US disclosed
EP-0960102-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN Du Pont Pharmaceuticals Company (US) 1999-12-01 EP disclosed
US-5886191-A ANTICOAGULANTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-23 US disclosed
WO-1998001428-A1 AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN DU PONT PHARMACEUTICALS COMPANY (US) 1998-01-15 WO disclosed