SCHEMBL7367744

SCHEMBL7367744

CCn1nc(-c2c(C(=O)O)cccc2-c2ccccc2)cc(Nc2cccc3c2ccc[n+]3[O-])c1=O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 14/20 0.45
TP53 P04637 1/20 0.38
FABP3 P05413 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
ADORA1 P30542 3/20 0.34
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051034 0.86 PDE4B (0.39) PDE4BADORA1ADORA2AADORA2B
SCHEMBL7320567 0.83 PDE4B (0.48) PDE4BADORA1ADORA2AADORA2B
SCHEMBL7367748 0.81 PDE4B (0.47) PDE4BTP53FABP3FABP4FABP5
SCHEMBL7308254 0.79 PDE4B (0.54) PDE4BADORA1ADORA2AADORA2B
SCHEMBL4058822 0.79 PDE4B (0.36) PDE4BTP53ADORA1ADORA2AADORA2B
SCHEMBL3031978 0.73 PDE4B (0.57) PDE4BTP53ADORA1
SCHEMBL3022288 0.68 PDE4B (0.47) PDE4BTP53ADORA1ADORA2AADORA2B
SCHEMBL3022169 0.68 PDE4B (0.47) PDE4BTP53
SCHEMBL3029571 0.67 PDE4B (0.49) PDE4BTP53
SCHEMBL4052027 0.67 PDE4B (0.54) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394998-A1 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3-yl)-biphenyl derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2011-12-14 EP disclosed