SCHEMBL7368433

SCHEMBL7368433

COc1ccc2c(c1)OC(=O)C(N)C2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KYAT1 Q16773 1/20 0.51
KYAT3 Q6YP21 1/20 0.51
AADAT Q8N5Z0 1/20 0.51
ALDH1A1 P00352 2/20 0.45
ACHE P22303 1/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
BACE1 P56817 1/20 0.42
CYP19A1 P11511 4/20 0.42
MAOB P27338 3/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.41
PPARG P37231 2/20 0.39
PPARA Q07869 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30373725 0.82 ALDH1A1 (0.45) KYAT1KYAT3AADATALDH1A1ACHE
SCHEMBL28990291 0.82 ALDH1A1 (0.45) KYAT1KYAT3AADATALDH1A1ACHE
SCHEMBL28999685 0.78 PPARG (0.48) ALDH1A1ACHEBACE1CYP19A1MAOB
SCHEMBL28555018 0.77 CYP19A1 (0.55) ALDH1A1CYP19A1MAOBCYP3A4MAPT
SCHEMBL14007732 0.76 ESR2 (0.43) ALDH1A1DRD2DRD3CA2CA5A
SCHEMBL14389073 0.76 ALDH1A1 (0.52) ALDH1A1CYP19A1MAOBCYP3A4MAPT
SCHEMBL12283677 0.74 PPARG (0.51) ALDH1A1BACE1CYP19A1MAOBMAPT
SCHEMBL28999667 0.73 PPARG (0.54) ALDH1A1BACE1MAOBMAPTPPARG
SCHEMBL10206132 0.73 ACHE (0.69) KYAT1KYAT3AADATACHEDRD2
SCHEMBL14495775 0.72 CA12 (0.54) ALDH1A1CA2CA5AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441974-A Phenyl amidines lactones useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-08-15 US disclosed
WO-1993012103-A1 PHENYL AMIDINES LACTONES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-06-24 WO disclosed