SCHEMBL7368439

SCHEMBL7368439

CCOC(=O)CN(CCCCc1ccc(N)cc1)c1cccc(C#N)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
PPARG P37231 3/20 0.39
F2 P00734 2/20 0.39
F10 P00742 2/20 0.39
PLG P00747 2/20 0.39
PLAT P00750 2/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
F7 P08709 2/20 0.39
PRSS3 P35030 2/20 0.39
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
FFAR1 O14842 2/20 0.38
LTA4H P09960 1/20 0.37
ALOX5 P09917 1/20 0.36
CYP1A2 P05177 1/20 0.36
GRM5 P41594 1/20 0.36
GFER P55789 1/20 0.36
SETD7 Q8WTS6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464051 0.93 PDCD1 (0.42) PDCD1CD274PPARGF2PRSS1
SCHEMBL7360601 0.87 KCNH2 (0.44) PDCD1CD274PPARGKDM4E
SCHEMBL7365136 0.86 F2 (0.42) PDCD1CD274PPARGF2F10
SCHEMBL7362325 0.85 FFAR1 (0.42) PPARGF2F10PLGPLAT
SCHEMBL7357492 0.85 FFAR1 (0.47) PPARGF2PRSS1PRSS2PRSS3
SCHEMBL7359452 0.85 PDCD1 (0.44) PDCD1CD274PPARGF2PRSS1
SCHEMBL7362903 0.83 F2 (0.56) F2F10PLGPLATPRSS1
SCHEMBL7361441 0.83 FFAR1 (0.44) PDCD1CD274PPARGFFAR1LTA4H
Trifluoroacetic Acid SCHEMBL7454966 0.79 F2 (0.59) F2F10PLGPLATPRSS1
SCHEMBL7362625 0.79 KCNH2 (0.46) PDCD1CD274KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892780-B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-11-20 EP disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed