SCHEMBL7368515

SCHEMBL7368515

NC(=O)c1cc(OCc2ccccc2)ccc1C[CH]C(=O)N(Cc1ccccc1)C1CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.44
MBTPS1 Q14703 3/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
KCNH2 Q12809 1/20 0.41
HTR2A P28223 1/20 0.41
TACR1 P25103 3/20 0.40
DCUN1D1 Q96GG9 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
UBE2M P61081 1/20 0.39
PRMT5 O14744 1/20 0.38
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370862 0.95 MBTPS1 (0.48) CACNA1BMBTPS1SLC6A2SLC6A4SLC6A3
SCHEMBL7368517 0.72 CACNA1B (0.47) CACNA1BMBTPS1SLC6A2SLC6A4SLC6A3
SCHEMBL5358933 0.72 PARP10 (0.51) SIRT2
SCHEMBL7375298 0.71 NPC1 (0.43) SIRT2
SCHEMBL6803013 0.70 SIRT2 (0.49) SIRT2
SCHEMBL6622412 0.70 DCUN1D1 (0.54) SLC6A2SLC6A4SLC6A3KCNH2TACR1
SCHEMBL3811903 0.69 DCUN1D1 (0.58) SLC6A2SLC6A4SLC6A3KCNH2TACR1
SCHEMBL5352876 0.69 SIRT2 (0.48) SIRT2
Hydrochloric Acid SCHEMBL21410210 0.68 DCUN1D1 (0.57) SLC6A2SLC6A4SLC6A3KCNH2TACR1
SCHEMBL6202628 0.68 HTR2A (0.51) SLC6A2SLC6A4SLC6A3KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed