SCHEMBL7368519

SCHEMBL7368519

O=C(O)CCNC(=O)C(Cc1ccc(-c2ccccc2)cc1)CP(=O)(O)O

nearest known ligand 0.85

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MMEL1 Q495T6 1/20 0.74
MME P08473 1/20 0.60
ACE P12821 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371290 1.00 MMEL1 (0.74) MMEL1MMEACE
SCHEMBL7371286 1.00 MMEL1 (0.74) MMEL1MMEACE
SCHEMBL7318461 0.92 ACE (0.70) MMEL1MMEACE
SCHEMBL7367811 0.92 ACE (0.70) MMEL1MMEACE
SCHEMBL7367809 0.92 ACE (0.70) MMEL1MMEACE
SCHEMBL10791111 0.91 ACE (0.68) MMEL1MMEACE
SCHEMBL10789074 0.91 ACE (0.68) MMEL1MMEACE
SCHEMBL8861591 0.87 MME (0.60) MMEL1MMEACE
SCHEMBL7367705 0.86 ACE (0.54) MMEL1MMEACE
SCHEMBL7361926 0.86 ACE (0.54) MMEL1MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0117429-B1 PHOSPHOROUS CONTAINING COMPOUNDS AS INHIBITORS OF ENKEPHALINASES SCHERING CORPORATION (US) 1987-09-02 EP claimed
EP-0117429-A1 Phosphorous containing compounds as inhibitors of enkephalinases SCHERING CORPORATION (US) 1984-09-05 EP claimed
CN-107257785-B (2S,4R) -5- (5 '-chloro-2' -fluorobiphenyl-4-yl) -4- (ethoxyoxalylamino) -2-hydroxymethyl-2-methylpentanoic acid as enkephalinase inhibitors 施万生物制药研发IP有限责任公司 2020-07-07 CN disclosed
EP-0117429-B1 PHOSPHOROUS CONTAINING COMPOUNDS AS INHIBITORS OF ENKEPHALINASES SCHERING CORPORATION (US) 1987-09-02 EP disclosed
EP-0117429-A1 Phosphorous containing compounds as inhibitors of enkephalinases SCHERING CORPORATION (US) 1984-09-05 EP disclosed