SCHEMBL7368657

SCHEMBL7368657

CCCCC(C(=O)O)N(C)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.45
MAPK1 P28482 1/20 0.45
SLC1A2 P43004 2/20 0.43
SLC1A1 P43005 2/20 0.43
SLC1A3 P43003 1/20 0.43
ACE2 Q9BYF1 1/20 0.40
GPR84 Q9NQS5 3/20 0.39
CA1 P00915 3/20 0.39
FFAR1 O14842 1/20 0.39
MAPT P10636 1/20 0.38
LCK P06239 1/20 0.38
PPARD Q03181 1/20 0.38
ZDHHC20 Q5W0Z9 1/20 0.38
ZDHHC2 Q9UIJ5 1/20 0.38
GRIK1 P39086 2/20 0.38
GRIK2 Q13002 2/20 0.38
CHRM1 P11229 1/20 0.37
AKR1A1 P14550 1/20 0.37
CHRM3 P20309 1/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23513672 0.92 GPR84 (0.50) CA2SLC1A2SLC1A1ACE2GPR84
SCHEMBL18510075 0.90 CA2 (0.50) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL22791880 0.82 CA2 (0.35) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL25847062 0.82 CA2 (0.35) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL11777790 0.82 GPR84 (0.55) CA2SLC1A2SLC1A1ACE2GPR84
SCHEMBL16585650 0.81 CA2 (0.50) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL2512194 0.81 CA2 (0.50) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL22384118 0.81 GSR (0.47)
SCHEMBL22384142 0.79 TP53 (0.33) CA2MAPK1SLC1A2SLC1A1SLC1A3
SCHEMBL22384047 0.78 CYP1A2 (0.50) SLC1A2SLC1A1SLC1A3GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed