SCHEMBL7369264

SCHEMBL7369264

O=C(O)C(Cc1ccc(C(F)(F)F)cc1)C(=O)c1cccnc1Oc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
FFAR1 O14842 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
PDE10A Q9Y233 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27514001 0.89 KMT2A (0.44) KMT2AKDM4EMEN1CYP1A2CYP2C19
SCHEMBL7367287 0.83 KMT2A (0.47) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL7374580 0.81 KMT2A (0.43) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL7372342 0.80 PDE10A (0.48) KMT2AKDM4EMEN1CYP1A2CYP2C19
SCHEMBL7405328 0.79 MAPK8 (0.55) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL7367980 0.78 KMT2A (0.54) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL7405885 0.77 KMT2A (0.45) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL2785360 0.77 TDP1 (0.54) KMT2AKDM4EMEN1CYP1A2CYP2C19
SCHEMBL7123489 0.74 GSK3B (0.49) FFAR1PPARGPPARA
SCHEMBL2779361 0.74 KMT2A (0.65) KMT2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed
EP-0663912-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1995-07-26 EP disclosed
EP-0663912-A4 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION. ABBOTT LAB (US) 1995-02-17 EP disclosed
WO-1994008992-A1 HETEROCYCLIC ETHER COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1994-04-28 WO disclosed