SCHEMBL7369538

SCHEMBL7369538

CC(C)CC(C(=O)O)N(C)Cc1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NR4A2 P43354 1/20 0.46
MME P08473 2/20 0.46
FPR2 P25090 1/20 0.43
MMP1 P03956 4/20 0.42
MMP3 P08254 4/20 0.42
CTSK P43235 1/20 0.41
MMP2 P08253 2/20 0.40
MMP7 P09237 2/20 0.40
MMP9 P14780 2/20 0.40
MMP8 P22894 1/20 0.40
MMP13 P45452 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EPHX1 P07099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7369241 1.00 PYCR1 (0.49) PYCR1MEN1KMT2ANR4A2MME
SCHEMBL7374458 0.86 NR4A2 (0.47) MEN1KMT2ANR4A2MMEMMP1
SCHEMBL7369868 0.86 NR4A2 (0.47) MEN1KMT2ANR4A2MMEMMP1
SCHEMBL7372235 0.86 NR4A2 (0.55) MEN1KMT2ANR4A2MMP1MMP3
SCHEMBL3039559 0.86 NR4A2 (0.55) MEN1KMT2ANR4A2MMP1MMP3
SCHEMBL7364441 0.85 HDAC1 (0.47) MEN1KMT2ANR4A2MMP1MMP3
SCHEMBL7364436 0.85 HDAC1 (0.47) MEN1KMT2ANR4A2MMP1MMP3
SCHEMBL7367268 0.85 TDP1 (0.47) MEN1KMT2ANR4A2HTT
SCHEMBL7372724 0.85 ALDH1A1 (0.47) NR4A2MMP1MMP3TSHRHTT
SCHEMBL7366036 0.85 TDP1 (0.47) MEN1KMT2ANR4A2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed