SCHEMBL7369982

SCHEMBL7369982

O=[N+]1N=CCc2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.33
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
MAOA P21397 1/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5706585 0.80 NOS3 (0.33) NOS3NOS1NOS2
SCHEMBL530203 0.77 HTR6 (0.33) HTR6
SCHEMBL7337539 0.71 CYP1A2 (0.35) NOS3NOS1NOS2MAOACYP1A2
SCHEMBL2461757 0.64 HTR6 (0.33) HTR6CYP1A2
Hydrochloric Acid SCHEMBL7370281 0.62 HTR6 (0.33) HTR6CYP1A2
SCHEMBL11611587 0.61 CYP1A2 (0.33) HTR6CYP1A2
SCHEMBL10677670 0.61 HTR6 (0.32) HTR6CYP1A2
SCHEMBL11880028 0.60 HTR6 (0.31) HTR6
SCHEMBL6672436 0.58 CYP1A2 (0.35) CYP1A2
SCHEMBL3649668 0.58 MAOB (0.38) NOS3NOS1NOS2MAOACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716954-A ANTIINFLAMMATORY AGENT, ANTIHISTAMINES, IMMUNOSUPPRESSION,AUTOIMMUNE DISEASES SYNTEX U.S.A. INC. (US) 1998-02-10 US disclosed
EP-0681582-A1 PYRAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF PHARMACIA & UPJOHN COMPANY (US) 1995-11-15 EP disclosed
EP-0612321-A1 PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1994-08-31 EP disclosed
WO-1993007146-A1 BENZO AND PYRIDO PYRIDAZINONE AND PYRIDAZINTHIONE COMPOUNDS WITH PDE IV INHIBITING ACTIVITY SYNTEX (U.S.A.) INC. (US) 1993-04-15 WO disclosed