SCHEMBL7370244

SCHEMBL7370244

NC(=O)c1cc(OCc2ccccc2)ccc1C[CH]C(=O)NCCNCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPHK2 Q9NRA0 1/20 0.47
SPHK1 Q9NYA1 1/20 0.47
SIRT2 Q8IXJ6 2/20 0.45
BCHE P06276 7/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
MAOB P27338 2/20 0.42
PARP10 Q53GL7 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PDCD1 Q15116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372540 0.91 NPC1 (0.47) SPHK2SPHK1SIRT2MAOBPARP10
SCHEMBL7373069 0.83 TDP1 (0.45) SIRT2PARP10MEN1KMT2A
SCHEMBL7367887 0.83 HTT (0.47) SIRT2
SCHEMBL7369351 0.82 NPC1 (0.48)
SCHEMBL7369285 0.81 EGFR (0.48)
SCHEMBL7369224 0.79 QPCT (0.54) KMT2A
SCHEMBL5358933 0.76 PARP10 (0.51) SIRT2MAOBPARP10KMT2A
SCHEMBL10957903 0.76 DRD4 (0.55) SPHK2SPHK1SIRT2MEN1KMT2A
SCHEMBL7375298 0.75 NPC1 (0.43) SPHK1SIRT2MAOBPARP10
Hydrochloric Acid SCHEMBL10959588 0.75 DRD4 (0.54) SPHK2SPHK1SIRT2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US claimed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO claimed
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed