SCHEMBL7370612

SCHEMBL7370612

COc1cccc2c(N)ccnc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.59
ADRA1D P25100 2/20 0.59
ADRA1A P35348 2/20 0.59
ADRA1B P35368 2/20 0.59
NR4A2 P43354 1/20 0.56
NSD2 O96028 1/20 0.50
CASP6 P55212 1/20 0.50
G6PD P11413 1/20 0.50
IDO1 P14902 2/20 0.47
MCHR1 Q99705 1/20 0.46
EP300 Q09472 1/20 0.46
KAT8 Q9H7Z6 1/20 0.46
PLAU P00749 1/20 0.45
NCF1 P14598 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
ALDH1A1 P00352 2/20 0.44
ADRA2B P18089 1/20 0.44
PTGS1 P23219 1/20 0.44
CYP3A4 P08684 1/20 0.44
HSP90AA1 P07900 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9181996 0.86 NSD2 (0.58) HTR1AADRA1DADRA1AADRA1BNR4A2
SCHEMBL11428540 0.83 NR4A2 (0.53) HTR1AADRA1DADRA1AADRA1BNR4A2
SCHEMBL1337689 0.80 HTR1A (0.61) HTR1AADRA1DADRA1AADRA1BG6PD
SCHEMBL30543156 0.79 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BNSD2
SCHEMBL2699726 0.79 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BNSD2
SCHEMBL7247375 0.79 NSD2 (0.54) HTR1AADRA1DADRA1AADRA1BNR4A2
SCHEMBL2178344 0.79 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BNR4A2
SCHEMBL4014412 0.79 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BNSD2
SCHEMBL31337072 0.79 HTR1A (0.59) HTR1AADRA1DADRA1AADRA1BNSD2
SCHEMBL24715854 0.78 HTR1A (0.55) HTR1AADRA1DADRA1AADRA1BPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410529-B1 DIETETICS; NON-INSULIN DEPENDENT DIABETES; SLEEP DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 2002-06-25 US disclosed
EP-1003737-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2000-05-31 EP disclosed
WO-1999009024-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS HFGAN72 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1999-02-25 WO disclosed
US-4218369-A FOR DYEING POLYACRYLONITRILE PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1980-08-19 US disclosed