SCHEMBL7370652

SCHEMBL7370652

CC(C)C[C@@H](C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCN1CCOCC1)N(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 18/20 0.61
MMP2 P08253 1/20 0.53
MMP9 P14780 1/20 0.53
MMP8 P22894 1/20 0.53
PSMB11 A5LHX3 1/20 0.52
PSMA7 O14818 1/20 0.52
PSMB1 P20618 1/20 0.52
PSMA1 P25786 1/20 0.52
PSMA2 P25787 1/20 0.52
PSMA3 P25788 1/20 0.52
PSMA4 P25789 1/20 0.52
PSMB8 P28062 1/20 0.52
PSMB9 P28065 1/20 0.52
PSMA5 P28066 1/20 0.52
PSMB4 P28070 1/20 0.52
PSMB6 P28072 1/20 0.52
PSMB5 P28074 1/20 0.52
PSMB10 P40306 1/20 0.52
PSMB3 P49720 1/20 0.52
PSMB2 P49721 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408154 0.93 CTSS (0.54) TACR2MMP9MMP8PSMB8PSMB9
SCHEMBL7398380 0.92 CTSS (0.53) TACR2PSMB8PSMB9PSMB5PSMB10
SCHEMBL7405180 0.92 TACR2 (0.57) TACR2MMP2MMP9MMP8PSMB11
SCHEMBL7344537 0.90 TACR2 (0.64) TACR2MMP2MMP9MMP8
SCHEMBL8193543 0.88 TACR2 (0.62) TACR2MMP2MMP9MMP8
SCHEMBL7345251 0.86 TACR2 (0.60) TACR2MMP2MMP9MMP8PSMB11
SCHEMBL7370096 0.86 TACR2 (0.60) TACR2MMP2MMP9MMP8PSMB11
SCHEMBL7401617 0.85 TACR2 (0.58) TACR2MMP2MMP9MMP8
SCHEMBL7446475 0.84 CTSS (0.51) TACR2PSMB8PSMB9PSMB5PSMB10
SCHEMBL7342593 0.84 TACR2 (0.58) TACR2PSMB11PSMA7PSMB1PSMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed