SCHEMBL7408154

SCHEMBL7408154

CC(C)C[C@@H](C(=O)N[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCCN1CCCC1)N(C)C

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.54
TACR2 P21452 7/20 0.51
CTSK P43235 2/20 0.49
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
CTSL P07711 1/20 0.47
MME P08473 1/20 0.46
ACE P12821 1/20 0.46
CPA1 P15085 1/20 0.46
ACE2 Q9BYF1 1/20 0.46
PSMB8 P28062 1/20 0.46
PSMB9 P28065 1/20 0.46
PSMB5 P28074 1/20 0.46
PSMB10 P40306 1/20 0.46
PSMB2 P49721 1/20 0.46
HTT P42858 1/20 0.46
PTPN1 P18031 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7398380 0.99 CTSS (0.53) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7370652 0.93 TACR2 (0.61) TACR2PSMB8PSMB9PSMB5PSMB10
SCHEMBL7446475 0.91 CTSS (0.51) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7401303 0.91 CTSS (0.50) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7399324 0.89 CTSS (0.48) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL8193256 0.89 CTSS (0.48) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7345872 0.88 CTSS (0.55) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL8193049 0.88 CTSS (0.48) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7337508 0.87 CTSS (0.55) CTSSTACR2CTSKITGB3ITGA2B
SCHEMBL7337619 0.87 CACNA1B (0.57) CTSSTACR2CTSKCTSLPSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117841-A USED TO TREAT STROKE, CEREBRAL ISCHEMIA, PAIN, HEAD TRAUMA OR EPILEPSY WARNER-LAMBERT COMPANY (US) 2000-09-12 US disclosed
WO-1998054123-A1 SUBSTITUTED PEPTIDYLAMINE CALCIUM CHANNEL BLOCKERS WARNER-LAMBERT COMPANY (US) 1998-12-03 WO disclosed