Benzene

Benzene

SCHEMBL7370712

C=C(C)C(=O)NN1CCNCC1.c1ccccc1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNAI3 P08754 1/20 0.41
GNAO1 P09471 1/20 0.41
GNAI1 P63096 1/20 0.41
ALDH1A1 P00352 4/20 0.36
SIGMAR1 Q99720 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 1/20 0.36
OPRD1 P41143 2/20 0.35
HTR6 P50406 2/20 0.33
GAA P10253 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTT P42858 2/20 0.32
ABCC1 P33527 1/20 0.31
CHRM5 P08912 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6853292 0.77 HTT (0.37) ALDH1A1KDM4EPOLBGAAL3MBTL1
SCHEMBL842713 0.75 HTT (0.40) ALDH1A1KDM4EPOLBGAAL3MBTL1
SCHEMBL1394575 0.74 GNAI3 (0.49) GNAI3GNAO1GNAI1ALDH1A1SIGMAR1
SCHEMBL7370715 0.73 KMT2A (0.42) ALDH1A1SIGMAR1KDM4EPOLBKMT2A
SCHEMBL27897257 0.73 CA12 (0.53) KMT2AGAAHTT
SCHEMBL29108006 0.72 GNAI3 (0.47) GNAI3GNAO1GNAI1ALDH1A1SIGMAR1
SCHEMBL3267951 0.72 GNAI3 (0.46) GNAI3GNAO1GNAI1ALDH1A1SIGMAR1
SCHEMBL1147606 0.72 CYP2D6 (0.45) POLBKMT2ARECQLBLML3MBTL1
SCHEMBL11443167 0.71 GNAI3 (0.42) GNAI3GNAO1GNAI1KDM4EPOLB
SCHEMBL717372 0.68 HTT (0.69) ALDH1A1SIGMAR1POLBOPRD1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280627-B1 DERIVATIVES OF N-SUBSTITUTED ALPHA-MERCAPTOMETHYL-BENZENE-PROPANAMIDE, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-04-21 EP disclosed
US-4839358-A ANALGESICS, ANTIDEPRESSANTS, ANTIANXIETY AGENTS ROUSSEL UCLAF (FR) 1989-06-13 US disclosed
EP-0280627-A2 Derivatives of N-substituted alpha-mercaptomethyl-benzene-propanamide, process for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-08-31 EP disclosed