SCHEMBL7371015

SCHEMBL7371015

NC(=O)N1CC[C@@](OC(=O)C(F)(F)F)(C(N)c2ccc3ccncc3c2)C1=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 1/20 0.33
PRMT3 O60678 1/20 0.32
CYP11B2 P19099 3/20 0.32
ACACB O00763 1/20 0.31
ACACA Q13085 1/20 0.31
ROCK2 O75116 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
AKT1 P31749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7368498 1.00 TPH1 (0.33) TPH1PRMT3CYP11B2ACACBACACA
SCHEMBL7385850 0.96 TPH1 (0.36) TPH1PRMT3CYP11B2ACACBACACA
SCHEMBL7375149 0.84 CYP11B2 (0.33) PRMT3CYP11B2
SCHEMBL7378268 0.69 CYP2A6 (0.38) PRMT3CYP11B2
SCHEMBL7374639 0.67 CYP11B2 (0.38) CYP11B2ROCK2
SCHEMBL7373348 0.64 CYP11B2 (0.38) CYP11B2ROCK2
Trifluoroacetic Acid SCHEMBL7376828 0.64 AKT1 (0.33) TPH1ROCK2AKT1
Trifluoroacetic Acid SCHEMBL7385179 0.64 DPP4 (0.38) TPH1AKT1
SCHEMBL7376941 0.64 CYP3A4 (0.31)
Trifluoroacetic Acid SCHEMBL7377917 0.63 DPP4 (0.39) TPH1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086099-A4 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARM PROD INC (US) 2002-01-02 EP claimed
EP-1086099-A1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS Aventis Pharmaceuticals Products Inc. (US) 2001-03-28 EP claimed
WO-1999062904-A1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-12-09 WO claimed
EP-1086099-A4 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARM PROD INC (US) 2002-01-02 EP disclosed
EP-1086099-A1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS Aventis Pharmaceuticals Products Inc. (US) 2001-03-28 EP disclosed
WO-1999062904-A1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-12-09 WO disclosed