SCHEMBL7372010

SCHEMBL7372010

CC(C)c1ccccc1Sc1c(O)cc(OCCN2CCN(C)CC2)oc1=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.36
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36
PRKDC P78527 1/20 0.36
HTR7 P34969 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
XDH P47989 2/20 0.35
P2RY12 Q9H244 1/20 0.35
DRD3 P35462 1/20 0.35
LTA4H P09960 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35
ITGAL P20701 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960964 0.80 ESR1 (0.40)
SCHEMBL6965961 0.79 BCHE (0.49) HRH3P2RY12LTA4HSIGMAR1
SCHEMBL6959993 0.79 ESR1 (0.41) XDHLTA4H
SCHEMBL6960575 0.79 BCHE (0.40)
SCHEMBL6965635 0.78 MEN1 (0.45) P2RY12SIGMAR1
SCHEMBL9040164 0.71 BCHE (0.34) SIGMAR1
SCHEMBL6961039 0.71 SMN1; SMN2 (0.46) L3MBTL1XDHHSP90AA1
SCHEMBL6954067 0.70 SIGMAR1 (0.36) HRH3DRD3SIGMAR1ITGB2ICAM1
SCHEMBL9038757 0.70 CYP2C9 (0.40)
SCHEMBL6963494 0.69 PTGES (0.43) L3MBTL1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed