SCHEMBL7373368

SCHEMBL7373368

CC[C@H](NC(=O)CN)C(=O)OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
TACR1 P25103 1/20 0.49
ACE P12821 1/20 0.48
CTSK P43235 1/20 0.48
MBTPS1 Q14703 1/20 0.47
ALDH1A1 P00352 2/20 0.46
CTSC P53634 2/20 0.46
LTA4H P09960 1/20 0.46
AOC3 Q16853 1/20 0.43
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30516239 0.87 ACE (0.62) POLBTACR1ACEMBTPS1CTSC
SCHEMBL18429658 0.87 ACE (0.62) POLBTACR1ACEMBTPS1CTSC
SCHEMBL18515876 0.87 ACE (0.62) POLBTACR1ACEMBTPS1CTSC
SCHEMBL3394167 0.86 CTSK (0.56) CTSKALDH1A1
SCHEMBL3394165 0.86 CTSK (0.56) CTSKALDH1A1
SCHEMBL30516234 0.86 CTSK (0.56) CTSKALDH1A1
SCHEMBL28288517 0.86 CTRB1 (0.51) POLBTACR1ACEMBTPS1ALDH1A1
Hydrochloric Acid SCHEMBL11526166 0.86 ACE (0.60) POLBTACR1ACEMBTPS1CTSC
Hydrochloric Acid SCHEMBL11604468 0.85 CTSK (0.55) CTSKALDH1A1
SCHEMBL26195471 0.84 CTSK (0.64) TACR1CTSKALDH1A1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810994-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-05-06 EP disclosed
US-5719162-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-02-17 US disclosed
US-5719144-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-02-17 US disclosed
EP-0810994-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1997-12-10 EP disclosed
US-5665723-A PIPERAZINE ISOINDOLE DERIVATIVES MERCK & CO., INC. (US) 1997-09-09 US disclosed
WO-1996026187-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-08-29 WO disclosed