SCHEMBL7373871

SCHEMBL7373871

CC(=O)Nc1cc(Cl)c(=O)n(C2=CC(C)(C)Oc3cnccc32)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.37
CCNC P24863 14/20 0.37
CDK8 P49336 14/20 0.37
HASPIN Q8TF76 13/20 0.37
CDK19 Q9BWU1 7/20 0.37
WEE1 P30291 1/20 0.35
ABL1 P00519 2/20 0.34
PDGFRB P09619 2/20 0.34
SRC P12931 2/20 0.34
PDGFRA P16234 2/20 0.34
MAPK14 Q16539 2/20 0.34
GRM1 Q13255 1/20 0.33
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377524 0.92 WEE1 (0.37) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7367507 0.89 AAK1 (0.37) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7290292 0.85 AAK1 (0.40) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7374768 0.85 CHUK (0.37) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7294332 0.84 CCNC (0.37) CCNCCDK8HASPINCDK19
SCHEMBL7291526 0.82 CCNC (0.40) CCNCCDK8HASPINCDK19
SCHEMBL7376992 0.81 AAK1 (0.35) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7376611 0.81 ALDH1A1 (0.38) CDK8CDK19WEE1ABL1PDGFRB
SCHEMBL7371406 0.81 CCNC (0.37) AAK1CCNCCDK8HASPINCDK19
SCHEMBL7374676 0.81 ALDH1A1 (0.38) WEE1ABL1PDGFRBSRCPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308792-B1 AZACHROMANE DERIVATIVES MERCK PATENT GmbH (DE) 1993-07-28 EP disclosed
US-4931454-A Azachroman derivatives with effects on the cardiovascular system MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-06-05 US disclosed