SCHEMBL7374152

SCHEMBL7374152

[CH2]c1cccc(-c2cc(N)on2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
BLM P54132 1/20 0.46
NOTUM Q6P988 3/20 0.41
RAB9A P51151 7/20 0.39
NPC1 O15118 6/20 0.39
KDR P35968 2/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAP4K4 O95819 1/20 0.36
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2E1 P05181 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2B6 P20813 1/20 0.34
HPGD P15428 2/20 0.33
HK1 P19367 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1787030 0.80 RAB9A (0.53) ALDH1A1MAPTKDM4EBLMNOTUM
SCHEMBL224856 0.79 RAB9A (0.61) ALDH1A1MAPTKDM4EBLMNOTUM
SCHEMBL7379131 0.79 RAB9A (0.47) ALDH1A1MAPTKDM4ENOTUMRAB9A
SCHEMBL1040166 0.79 CHEK1 (0.49) ALDH1A1MAPTKDM4EBLMRAB9A
SCHEMBL16826106 0.79 NOTUM (0.64) ALDH1A1MAPTKDM4EBLMNOTUM
SCHEMBL16826099 0.79 KDM4E (0.51) ALDH1A1MAPTKDM4EBLMNOTUM
SCHEMBL7372548 0.76 RORC (0.41) MAPTNOTUMRAB9ANPC1MEN1
SCHEMBL29615077 0.75 GRM5 (0.50) NOTUMMAP4K4
SCHEMBL22653460 0.75 NPC1 (0.54) ALDH1A1MAPTKDM4ERAB9ANPC1
SCHEMBL7375026 0.75 RAB9A (0.38) NOTUMRAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO claimed
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed
WO-1997008150-A1 SUBSTITUTED CYCLIC UREAS AND DERIVATIVES THEREOF USEFUL AS RETROVIRAL PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-06 WO disclosed