SCHEMBL7375802

SCHEMBL7375802

Cc1cccc2c(=O)cc(-c3c(O)ccc4ccccc34)oc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.55
CYP3A4 P08684 2/20 0.54
TSHR P16473 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A1 P04798 11/20 0.52
CYP1B1 Q16678 11/20 0.52
CYP1A2 P05177 10/20 0.52
CSNK2A2 P19784 2/20 0.52
CSNK2B P67870 2/20 0.52
CSNK2A1 P68400 2/20 0.52
PSMD14 O00487 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
CYP19A1 P11511 3/20 0.49
PRKDC P78527 2/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
ABCB1 P08183 2/20 0.49
ABCC1 P33527 2/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
PDE5A O76074 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15676498 0.79 CYP3A4 (0.67) CYP3A4TSHRCYP2C19CYP1A1CYP1B1
SCHEMBL4649417 0.75 CYP1B1 (0.63) CYP3A4TSHRCYP2C19CYP1A1CYP1B1
SCHEMBL7380906 0.74 CYP3A4 (0.64) MCL1CYP3A4TSHRCYP2C19CYP1A1
SCHEMBL14708624 0.71 MCL1 (1.00) MCL1CYP3A4TSHRCYP2C19CYP1A1
SCHEMBL12023067 0.71 CYP1A2 (0.52) TSHRCYP2C19CYP1A2TDP1KDM4E
SCHEMBL5432584 0.70 ALOX5 (0.57) CYP3A4CYP2C19TDP1TP53CYP2D6
SCHEMBL1319784 0.69 PRKDC (0.55) MCL1CYP3A4CYP2C19CYP1A1CYP1B1
SCHEMBL29677981 0.69 PRKDC (0.55) MCL1CYP3A4CYP2C19CYP1A1CYP1B1
SCHEMBL7374618 0.68 ALDH1A1 (0.82) CYP3A4TSHRCYP2C19CYP1A1CYP1B1
SCHEMBL12023086 0.68 ALDH1A1 (0.48) TSHRCYP2C19CYP1A2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115718-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000017184-A1 HYDROXYFLAVONE DERIVATIVES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI CHEMICAL CORPORATION (JP) 2000-03-30 WO disclosed