SCHEMBL7375883

SCHEMBL7375883

COC(=O)[C@H](CC(C)C)NC(=O)OCc1cccnc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.58
CTSB P07858 4/20 0.58
CTSK P43235 10/20 0.55
CYP3A4 P08684 1/20 0.53
CTSS P25774 3/20 0.52
CAPN1 P07384 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578032 0.90 CTSL (0.60) CTSLCTSBCTSKCYP3A4CTSS
SCHEMBL27497095 0.90 CTSL (0.60) CTSLCTSBCTSKCYP3A4CTSS
Lithium SCHEMBL7162098 0.89 CTSL (0.59) CTSLCTSBCTSKCYP3A4CTSS
SCHEMBL7162081 0.89 CTSL (0.59) CTSLCTSBCTSKCYP3A4CTSS
Lithium Ion SCHEMBL7162088 0.88 CTSL (0.56) CTSLCTSBCTSKCYP3A4CTSS
SCHEMBL27563904 0.85 CTSK (0.56) CTSLCTSBCTSKCTSSCAPN1
SCHEMBL7159540 0.85 CTSK (0.56) CTSLCTSBCTSKCTSSCAPN1
SCHEMBL14609392 0.84 CTSK (0.74) CTSLCTSBCTSKCTSSCAPN1
SCHEMBL13611959 0.84 CTSK (0.74) CTSLCTSBCTSKCTSSCAPN1
SCHEMBL3978105 0.84 CTSK (0.74) CTSLCTSBCTSKCTSSCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934291-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-08-11 EP disclosed
EP-0934291-A4 SMITHKLINE BEECHAM CORP (US) 1999-08-11 EP disclosed
WO-1997016433-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1997-05-09 WO disclosed