SCHEMBL7375936

SCHEMBL7375936

N#Cc1ccc(F)cc1.[Ar]

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.61
TP53 P04637 1/20 0.61
MAOA P21397 2/20 0.55
MAOB P27338 2/20 0.55
PTGS1 P23219 1/20 0.52
CYP2A6 P11509 2/20 0.50
CA2 P00918 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CA12 O43570 1/20 0.50
CA3 P07451 1/20 0.50
CA6 P23280 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
TSHR P16473 1/20 0.48
KIF11 P52732 1/20 0.44
NSD2 O96028 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
MMP3 P08254 1/20 0.44
ENPP2 Q13822 1/20 0.44
CYP11B1 P15538 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL39936 0.97
SCHEMBL12444126 0.97
Water SCHEMBL28049243 0.97 KDM4E (0.64) KDM4ETP53MAOAMAOBPTGS1
SCHEMBL28783861 0.94 KDM4E (0.61) KDM4ETP53MAOAMAOBPTGS1
SCHEMBL28251780 0.94 KDM4E (0.61) KDM4ETP53MAOAMAOBPTGS1
Hydrochloric Acid SCHEMBL30942103 0.94 KDM4E (0.61) KDM4ETP53MAOAMAOBPTGS1
SCHEMBL7929151 0.89 MMP3 (0.58) KDM4ETP53MAOAMAOBPTGS1
SCHEMBL15934230 0.89 KDM4E (0.57) KDM4ETP53MAOAMAOBPTGS1
SCHEMBL28311757 0.87 KDM4E (0.55) KDM4ETP53MAOAMAOBPTGS1
Ammonia Solution, Strong SCHEMBL3940933 0.85 KDM4E (0.53) KDM4ETP53MAOAMAOBPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773463-A DECALCIFICATION OF BRAIN DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 1998-06-30 US disclosed
EP-0711272-A1 INDANE AND TETRAHYDRONAPHTHALENE DERIVATIVES AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-05-15 EP disclosed
WO-1995004028-A1 INDANE AND TETRAHYDRONAPHTHALENE DERIVATIVES AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-02-09 WO disclosed