SCHEMBL7377358

SCHEMBL7377358

O=C[C@H](Cc1ccccc1)NC(=O)c1cccc(C(=O)c2ccccc2)c1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 10/20 0.70
ATM Q13315 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CTRB1 P17538 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786975 1.00 CAPN1 (0.70) CAPN1ATMTDP1L3MBTL1CTRB1
SCHEMBL7789383 0.90 CAPN1 (0.75) CAPN1CTRB1
SCHEMBL7374424 0.90 CAPN1 (0.75) CAPN1CTRB1
SCHEMBL7378642 0.87 CAPN1 (0.74) CAPN1CTRB1
SCHEMBL40781 0.87 CAPN1 (0.74) CAPN1CTRB1
SCHEMBL22098385 0.85 CAPN1 (0.61) CAPN1
SCHEMBL7787032 0.82 CAPN1 (1.00) CAPN1
SCHEMBL7376183 0.82 CAPN1 (1.00) CAPN1
SCHEMBL24862929 0.80 ALDH1A1 (0.60) CAPN1
SCHEMBL7789884 0.80 ROCK2 (0.57) ATMTDP1L3MBTL1CTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
EP-0944584-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998023581-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-04 WO disclosed