SCHEMBL7377481

SCHEMBL7377481

C(#Cc1ccccn1)C1=CCCC2CCCCC12

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 17/20 0.50
CYP1A2 P05177 8/20 0.50
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419198 0.71 GRM5 (0.59) GRM5CYP1A2
SCHEMBL352291 0.70 GRM5 (0.65) GRM5CYP1A2KCNH2
SCHEMBL4807933 0.68 GRM5 (0.96) GRM5CYP1A2KCNH2
SCHEMBL7377478 0.68 GRM5 (0.57) GRM5CYP1A2
SCHEMBL4856019 0.67 GRM5 (0.57) GRM5CYP1A2
SCHEMBL4863469 0.67 GRM5 (0.57) GRM5CYP1A2
Methyl Alcohol SCHEMBL28902013 0.66 GRM5 (0.67) GRM5CYP1A2KCNH2
SCHEMBL4860791 0.65 GRM5 (0.45) GRM5CYP1A2KCNH2
SCHEMBL7385260 0.64 GRM5 (0.54) GRM5CYP1A2
SCHEMBL4860119 0.64 GRM5 (0.97) GRM5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed