SCHEMBL7377900

SCHEMBL7377900

O=C(OC(=O)[C@@H]1CCCN1)C(CCS)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.47
FOLH1 Q04609 3/20 0.41
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
CPA3 P15088 1/20 0.39
ELANE P08246 1/20 0.38
TSHR P16473 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 1/20 0.37
SLC6A2 P23975 3/20 0.37
SLC6A3 Q01959 3/20 0.37
SLC6A4 P31645 2/20 0.37
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381712 0.91 CTSC (0.48) CTSCFOLH1HTR2CHTR2BCPA3
SCHEMBL11560126 0.89 CPA3 (0.49) CTSCHTR2CHTR2BCPA3ELANE
SCHEMBL11557590 0.87 CTSC (0.45) CTSCHTR2CHTR2BCPA3ELANE
SCHEMBL11556969 0.86 CPA1 (0.50) CTSCFOLH1HTR2CHTR2BCPA3
SCHEMBL11561006 0.85 CTSC (0.46) CTSCFOLH1HTR2CHTR2BCPA3
SCHEMBL11560751 0.85 CTSC (0.46) CTSCHTR2CHTR2BCPA3TSHR
SCHEMBL11558104 0.84 CTSC (0.47) CTSCHTR2CHTR2BCPA3ELANE
SCHEMBL7381470 0.83 CTSC (0.42) CTSCHTR2CHTR2BELANETSHR
SCHEMBL11559645 0.82 CTSC (0.47) CTSCHTR2CHTR2BTSHRCYP3A4
SCHEMBL11561516 0.82 LTA4H (0.48) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed
US-4046889-A HYPOTENSIVE AGENTS, ENZYME INHIBITORS, ANGIOTENSIN CONVERSION E. R. SQUIBB & SONS, INC. (US) 1977-09-06 US disclosed