SCHEMBL7378366

SCHEMBL7378366

CCOC(=O)CCc1cc(-c2ccccc2)n(-c2ccc3[nH]c(CNc4ccc(C#N)cc4)nc3c2C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.37
ALDH1A1 P00352 3/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
CYP1A2 P05177 1/20 0.35
TSHR P16473 1/20 0.35
ALOX5 P09917 3/20 0.35
SLC16A3 O15427 3/20 0.35
SLC16A1 P53985 3/20 0.35
PTGS1 P23219 2/20 0.34
TGFBR1 P36897 4/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378652 0.93 ALDH1A1 (0.38) MAPTALDH1A1NPC1LMNAMAPK1
Hydrochloric Acid SCHEMBL7379211 0.91 RXRA (0.44) MAPTALDH1A1NPC1LMNAMAPK1
SCHEMBL7379560 0.81 KLK1 (0.38) MAPTALDH1A1NPC1LMNAMAPK1
SCHEMBL7378005 0.81 KLK5 (0.42) MAPTALDH1A1NPC1LMNAMAPK1
Hydrochloric Acid SCHEMBL7380734 0.81 KLK1 (0.37) MAPTALDH1A1NPC1LMNAMAPK1
Hydrochloric Acid SCHEMBL7373824 0.80 KLK5 (0.42) MAPTALDH1A1NPC1LMNAMAPK1
SCHEMBL7379565 0.80 KLK1 (0.44) MAPTALDH1A1NPC1LMNAMAPK1
SCHEMBL7372469 0.76 KLK1 (0.46) MAPTALDH1A1NPC1LMNAMAPK1
SCHEMBL7383225 0.74 KLK1 (0.40) CYP1A2TSHR
SCHEMBL7394949 0.72 ALDH1A1 (0.43) MAPTALDH1A1NPC1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000050419-A1 SUBSTITUTED BICYCLIC HETEROCYCLES AND THE USE THEREOF AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-08-31 WO disclosed