SCHEMBL7378809

SCHEMBL7378809

NN=CNc1cccc(C(=O)Nc2ccc(CC(C(=O)O)c3ccccc3)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.50
ITGB3 P05106 10/20 0.48
ITGA2B P08514 10/20 0.48
ITGAV P06756 9/20 0.48
ITGB1 P05556 9/20 0.48
ITGB5 P18084 7/20 0.48
ALDH1A1 P00352 1/20 0.45
FFAR1 O14842 2/20 0.45
MEN1 O00255 1/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.45
KMT2A Q03164 1/20 0.45
ITGA4 P13612 2/20 0.45
MMP9 P14780 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7803105 0.87 ITGB3 (0.49) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7381611 0.86 ITGB3 (0.64) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7377112 0.86 ITGB3 (0.55) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7381617 0.86 ITGB3 (0.64) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7378200 0.86 ITGB3 (0.56) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7378198 0.86 ITGB3 (0.56) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7378626 0.85 ITGB3 (0.51) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7864788 0.84 SIRT2 (0.44) NR1H4ALDH1A1
SCHEMBL7457847 0.84 MEN1 (0.51) NR1H4ITGB3ITGA2BITGAVITGB1
SCHEMBL7457481 0.84 NR1H4 (0.67) NR1H4ITGB3ITGA2BITGAVITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-B1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2002-02-06 EP claimed
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed