SCHEMBL7378973

SCHEMBL7378973

CC(S)C(=O)OC(=O)[C@@H]1CCCN1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
PRCP P42785 1/20 0.35
DPP4 P27487 4/20 0.34
DPP7 Q9UHL4 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
DPP8 Q6V1X1 2/20 0.33
DPP9 Q86TI2 2/20 0.33
SCN4A P35499 1/20 0.33
TLR2 O60603 2/20 0.33
ELANE P08246 1/20 0.33
FAP Q12884 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11379805 0.87 NOS2 (0.33) NOS2NOS3NOS1PRCPDPP4
SCHEMBL9592134 0.86 NOS2 (0.37) NOS2NOS3NOS1PRCPDPP4
SCHEMBL1740647 0.85 NOS2 (0.36) NOS2NOS3NOS1PRCPDPP4
Hydrochloric Acid SCHEMBL6026726 0.85 NOS2 (0.36) NOS2NOS3NOS1PRCPDPP4
SCHEMBL28695544 0.85 NOS2 (0.36) NOS2NOS3NOS1PRCPDPP4
SCHEMBL27646576 0.83 NOS2 (0.39) NOS2NOS3NOS1PRCPDPP4
SCHEMBL20839948 0.83 NOS2 (0.35) NOS2NOS3NOS1PRCPDPP4
SCHEMBL499450 0.83 NOS2 (0.39) NOS2NOS3NOS1PRCPDPP4
SCHEMBL15210886 0.83 NOS2 (0.39) NOS2NOS3NOS1PRCPDPP4
SCHEMBL11434311 0.83 CYP3A4 (0.33) NOS2NOS3NOS1PRCPDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4745124-A THIO/ESTER PEPTIDES UNIVERSITY OF MIAMI (US) 1988-05-17 US disclosed
US-4692459-A SULFUR CONTAINING AMINO ACID DERIVATIVES, ANGIOTENSIN INHIBITOR UNIVERSITY OF MIAMI (US) 1987-09-15 US disclosed
EP-0035383-B1 ANGIOTENSIN CONVERTING ENZYME INHIBITORS UNIVERSITY OF MIAMI (US) 1984-05-30 EP disclosed
EP-0035383-A1 Angiotensin converting enzyme inhibitors UNIVERSITY OF MIAMI (US) 1981-09-09 EP disclosed
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed
US-4046889-A HYPOTENSIVE AGENTS, ENZYME INHIBITORS, ANGIOTENSIN CONVERSION E. R. SQUIBB & SONS, INC. (US) 1977-09-06 US disclosed