SCHEMBL7379693

SCHEMBL7379693

COc1cc2c(cc1OC)C(OS(=O)(=O)C(F)(F)F)=CCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
MAOA P21397 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ABCB1 P08183 1/20 0.37
CA7 P43166 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19127634 0.83 MPO (0.51) KDM4EALDH1A1MAPTKMT2AGLA
SCHEMBL30940171 0.83 MPO (0.51) KDM4EALDH1A1MAPTKMT2AGLA
SCHEMBL5364953 0.82 DRD2 (0.31) DRD2
SCHEMBL5847372 0.82 MPO (0.44) ALDH1A1MAOADRD2MPOABHD6
SCHEMBL29756733 0.82 MPO (0.44) ALDH1A1MAOADRD2MPOABHD6
SCHEMBL19616624 0.78 METAP1 (0.37) MAPTKMT2AMEN1DRD2
SCHEMBL18845471 0.78 METAP1 (0.37) MAPTKMT2AMEN1DRD2MPO
SCHEMBL2303778 0.77 MEN1 (0.41) KDM4EALDH1A1GAAMAPTMAOA
SCHEMBL4809246 0.77 MEN1 (0.41) KDM4EALDH1A1GAAMAPTMAOA
SCHEMBL5379087 0.77 KDM4C (0.39) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed