SCHEMBL7379989

SCHEMBL7379989

COc1ccc(NCC(F)(F)c2ccc(Cl)cc2CN)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.42
GAA P10253 6/20 0.42
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 6/20 0.36
APP P05067 1/20 0.36
KDM4E B2RXH2 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
HPGD P15428 1/20 0.36
KCNH2 Q12809 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381283 0.82 MAPT (0.41) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL6926332 0.71 KMT2A (0.42) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL5294889 0.69 GAA (0.67) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL1196343 0.69 NOS3 (0.47) MAPTMEN1KMT2ATDP1HPGD
SCHEMBL6920258 0.68 MEN1 (0.46) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL6921465 0.68 ALDH1A1 (0.43) MAPTGAAMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL4496671 0.67 NOS3 (0.46) MAPTMEN1KMT2ATDP1HPGD
SCHEMBL15114279 0.67 GAA (0.64) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL18235948 0.67 MAPT (0.55) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL18235922 0.66 GAA (0.62) MAPTGAAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002050056-A1 BENZYLAMINE DERIVATIVES AND THEIR USE AS THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-06-27 WO disclosed