SCHEMBL7380340

SCHEMBL7380340

CN(C)C1(NC(=O)c2cccc(NC(=N)N)c2)C=CC=CC1CCC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.37
ITGA2B P08514 5/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PARP1 P09874 1/20 0.35
PARP10 Q53GL7 1/20 0.35
KCNK3 O14649 1/20 0.35
KCNK9 Q9NPC2 1/20 0.35
ROCK2 O75116 2/20 0.34
PLK4 O00444 1/20 0.34
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34
CHUK O15111 1/20 0.34
DAPK3 O43293 1/20 0.34
JAK2 O60674 1/20 0.34
PAK4 O96013 1/20 0.34
CHEK2 O96017 1/20 0.34
CDK1 P06493 1/20 0.34
PIM1 P11309 1/20 0.34
PRKACA P17612 1/20 0.34
FGFR3 P22607 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7372592 0.86 ITGB3 (0.39) ITGB3ITGA2BSMN1; SMN2PARP1PARP10
SCHEMBL7348070 0.79 HTT (0.38) ITGB3ITGA2BSMN1; SMN2PARP1PARP10
SCHEMBL7340322 0.77 EPHX2 (0.37) ITGB3ITGA2BSMN1; SMN2PARP1PARP10
SCHEMBL7343615 0.70 SMN1; SMN2 (0.38) ITGB3ITGA2BSMN1; SMN2PARP1PARP10
SCHEMBL7379949 0.69 ITGB3 (0.51) ITGB3ITGA2BSMN1; SMN2KCNK3KCNK9
SCHEMBL7380345 0.68 KCNK3 (0.50) ITGB3ITGA2BSMN1; SMN2KCNK3KCNK9
SCHEMBL8441143 0.68 PARP1 (0.40) ITGB3ITGA2BPARP1PARP10ROCK2
SCHEMBL7340450 0.68 HTT (0.37) ITGB3ITGA2BSMN1; SMN2EPHX2MEN1
SCHEMBL8500073 0.68 MAPT (0.49) ITGB3ITGA2BSMN1; SMN2ITGAVKMT2A
SCHEMBL7347196 0.67 HTT (0.37) ITGB3ITGA2BSMN1; SMN2PARP1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed