SCHEMBL7380404

SCHEMBL7380404

Nc1cc(-c2ccc(Cl)cc2Cl)nc(N)n1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.75
HSP90AB1 P08238 5/20 0.75
LMNA P02545 1/20 0.53
KDM4E B2RXH2 2/20 0.50
RAB9A P51151 2/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
PTPN1 P18031 1/20 0.49
BACE1 P56817 1/20 0.48
AGPAT2 O15120 3/20 0.48
HTR2B P41595 1/20 0.47
PDE4D Q08499 1/20 0.47
MGAM O43451 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
AMY1A P0DUB6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944846 0.86 HSP90AB1 (1.00) HSP90AA1HSP90AB1LMNAKDM4ERAB9A
SCHEMBL7375654 0.80 HSP90AA1 (0.74) HSP90AA1HSP90AB1LMNAKDM4EMAPT
SCHEMBL15757500 0.79 HSP90AA1 (0.66) HSP90AA1HSP90AB1LMNAPTPN1AGPAT2
SCHEMBL7383642 0.79 SCN2A (0.49) HSP90AA1HSP90AB1AGPAT2HTR2BPDE4D
SCHEMBL1759878 0.77 MAPT (0.72) HSP90AA1HSP90AB1LMNAKDM4ERAB9A
SCHEMBL3602925 0.77 HSP90AA1 (0.51) HSP90AA1HSP90AB1LMNAKDM4ERAB9A
SCHEMBL7379292 0.76 KDM4E (0.62) HSP90AA1HSP90AB1KDM4ERAB9ANPC1
SCHEMBL9566485 0.76 HTR2B (0.72) HSP90AA1HSP90AB1LMNAKDM4ERAB9A
SCHEMBL6049475 0.74 HSP90AB1 (0.59) HSP90AA1HSP90AB1LMNAKDM4ERAB9A
SCHEMBL7382138 0.74 NUDT1 (0.66) HSP90AA1HSP90AB1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP claimed
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed