SCHEMBL7375654

SCHEMBL7375654

Nc1cc(-c2ccccc2Cl)nc(N)n1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 7/20 0.74
HSP90AB1 P08238 6/20 0.74
MAPK14 Q16539 2/20 0.52
CHRNA7 P36544 1/20 0.51
NUDT1 P36639 2/20 0.49
ADORA2A P29274 3/20 0.47
ADORA1 P30542 3/20 0.47
PTPN1 P18031 1/20 0.46
BACE1 P56817 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAOB P27338 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPK10 P53779 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7382138 0.86 NUDT1 (0.66) HSP90AA1HSP90AB1MAPK14CHRNA7NUDT1
SCHEMBL3950560 0.85 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAPK14CHRNA7NUDT1
SCHEMBL18672484 0.83 HSP90AA1 (0.53) HSP90AA1HSP90AB1MAPK14NUDT1
SCHEMBL7377883 0.80 DHFR (0.49) HSP90AA1HSP90AB1ADORA2AADORA1MEN1
SCHEMBL7380404 0.80 HSP90AA1 (0.75) HSP90AA1HSP90AB1PTPN1BACE1KDM4E
SCHEMBL20400592 0.80 HSP90AA1 (0.66) HSP90AA1HSP90AB1MAPK14CHRNA7NUDT1
SCHEMBL30400452 0.80 HSP90AA1 (0.66) HSP90AA1HSP90AB1MAPK14CHRNA7NUDT1
Hydrochloric Acid SCHEMBL5749719 0.79 DHFR (0.47) HSP90AA1HSP90AB1ADORA2AADORA1MEN1
SCHEMBL15757710 0.78 NUDT1 (0.78) HSP90AA1HSP90AB1MAPK14CHRNA7NUDT1
SCHEMBL29044794 0.78 NUDT1 (0.50) HSP90AA1HSP90AB1MAPK14NUDT1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP claimed
EP-0459830-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed