SCHEMBL7380480

SCHEMBL7380480

CCOC(=O)C(=O)c1ccc(OC2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.59
CHEK2 O96017 1/20 0.53
PDE4D Q08499 3/20 0.52
PDE4A P27815 2/20 0.52
PDE4B Q07343 2/20 0.52
PDE4C Q08493 2/20 0.52
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7388684 0.94 GPR119 (0.52) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL7389633 0.94 GPR119 (0.52) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL1375168 0.89 GPR119 (0.61) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL7392069 0.85 CHEK2 (0.55) GPR119CHEK2KMT2A
SCHEMBL1376438 0.84 PDE4D (0.56) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL1375476 0.84 GPR119 (0.60) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL20046236 0.83 GPR119 (0.55) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL6192490 0.82 GPR119 (0.62) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL1649132 0.82 GPR119 (0.64) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL3345205 0.82 GPR119 (0.64) GPR119CHEK2PDE4DPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962695-A ANTICOAGULANT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1999-10-05 US disclosed
US-5620991-A ANTICOAGULANTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-04-15 US disclosed
US-5576343-A ANTICOAGULANTS; BLOOD-COAGULATION FACTOR X INHIBITORS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-11-19 US disclosed
EP-0540051-B1 Aromatic amidine derivatives and salts thereof DAIICHI SEIYAKU CO (JP) 1996-04-03 EP disclosed
EP-0540051-A1 Aromatic amidine derivatives and salts thereof DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-05-05 EP disclosed