SCHEMBL7388684

SCHEMBL7388684

CCOC(=O)C(=O)c1ccc(O[C@H]2CCN(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.52
USP30 Q70CQ3 1/20 0.49
CHEK2 O96017 2/20 0.49
PDE4D Q08499 3/20 0.46
PDE4A P27815 2/20 0.46
PDE4B Q07343 2/20 0.46
PDE4C Q08493 2/20 0.46
KMT2A Q03164 1/20 0.44
PIK3CD O00329 3/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7389633 1.00 GPR119 (0.52) GPR119USP30CHEK2PDE4DPDE4A
SCHEMBL7380480 0.94 GPR119 (0.59) GPR119CHEK2PDE4DPDE4APDE4B
SCHEMBL7379041 0.88 GPR119 (0.52) GPR119USP30CHEK2PDE4DPDE4A
SCHEMBL1375168 0.84 GPR119 (0.61) GPR119USP30CHEK2PDE4DPDE4A
SCHEMBL5544755 0.83 USP30 (0.58) GPR119USP30CHEK2KMT2APIK3CD
SCHEMBL5545000 0.83 USP30 (0.58) GPR119USP30CHEK2KMT2APIK3CD
SCHEMBL240368 0.83 USP30 (0.58) GPR119USP30CHEK2KMT2APIK3CD
SCHEMBL6188750 0.83 GPR119 (0.54) GPR119USP30PIK3CDPOLB
SCHEMBL7386960 0.83 GPR119 (0.52) GPR119USP30CHEK2PIK3CD
SCHEMBL3911512 0.83 GPR119 (0.52) GPR119USP30CHEK2KMT2APIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962695-A ANTICOAGULANT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1999-10-05 US disclosed
US-5866577-A AN ANTICOAGULANT AGENT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1999-02-02 US disclosed
US-5620991-A ANTICOAGULANTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-04-15 US disclosed
US-5576343-A ANTICOAGULANTS; BLOOD-COAGULATION FACTOR X INHIBITORS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-11-19 US disclosed
EP-0540051-B1 Aromatic amidine derivatives and salts thereof DAIICHI SEIYAKU CO (JP) 1996-04-03 EP disclosed
EP-0540051-A1 Aromatic amidine derivatives and salts thereof DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-05-05 EP disclosed